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Agonist activity at full length human ERbeta receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:13 Active, 5 Activity ≤ 1 nM, 13 Activity ≤ 1 µM, 13 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at full length human ERalpha receptor assessed as transcriptional activity incubated for 22 to 24 hrs by cell based luciferase reporter gene assay
Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested
Displacement of fluormone from GST-tagged ERbeta receptor LBD (unknown origin) measured after 60 mins by TR-FRET competitive binding assay
Assay data:14 Active, 5 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 14 Tested
BK Channel Variant Modulator Selectivity Assay
Assay data:286 Active, 904 Activity ≤ 1 nM, 951 Activity ≤ 1 µM, 951 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Displacement of 17beta-[3H]estradiol from rabbit uterine estrogen receptor after 16 to 18 hrs by liquid scintillation counting
Assay data:4 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway: Summary
Assay data:589 Active, 16 Activity ≤ 1 nM, 99 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
DRUGMATRIX: Estrogen ERalpha radioligand binding (ligand: [3H] Estradiol)
Assay data:20 Active, 5 Activity ≤ 1 nM, 16 Activity ≤ 1 µM, 871 Tested
qHTS assay for small molecule agonists of estrogen receptor alpha signaling
Assay data:88 Active, 2 Activity ≤ 1 nM, 43 Activity ≤ 1 µM, 2858 Tested
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