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PDE SPA Enzyme Inhibition Assay from Article 10.1021/bi049868i: "Crystal structure of human phosphodiesterase 3B: atomic basis for substrate and inhibitor specificity."
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human His-tagged PDE3B catalytic domain expressed in Escherichia coli BL21(DE3) pLysS cells
Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB
Assay data:3598 Active, 421 Activity ≤ 1 nM, 2233 Activity ≤ 1 µM, 3598 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
qHTS for Inhibitors of binding or entry into cells for Lassa Virus
Assay data:3699 Active, 99 Activity ≤ 1 nM, 6304 Activity ≤ 1 µM, 300904 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS Validation Assay to Find Inhibitors of Chronic Active B-Cell Receptor Signaling
Assay data:6 Active, 41 Activity ≤ 1 µM, 1280 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
In vitro vascular relaxation in canine mesenteric veins precontracted with phenylephrine.
Assay data:20 Active, 10 Activity ≤ 1 µM, 21 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Antagonist binding of L-N6-phenyl-isopropyl)-[3H]adenosine to rat brain
Assay data:5 Active, 4 Activity ≤ 1 µM, 6 Tested
Antagonist binding of 2-chloro-[3H]-adenosine to rat brain
Assay data:7 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 8 Tested
Evaluated for Ca++ dependent phosphodiesterase activity.
Assay data:1 Active, 1 Activity ≤ 1 µM, 6 Tested
qHTS Assay for Lipid Storage Modulators
Assay data:19 Active, 2 Activity ≤ 1 nM, 490 Activity ≤ 1 µM, 8868 Tested
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