Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Cytochrome P450 family 3 subfamily A member 7 (CYP3A7) small molecule antagonists: luciferase cell-based qHTS assay
Assay data:2481 Active, 355 Activity ≤ 1 µM, 5246 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Depositor
Binding affinity towards human OPRM1 in an in vitro assay with cellular components measured by scintillation counting
Assay data:60 Active, 9 Activity ≤ 1 µM, 766 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity towards human PGR in an in vitro assay with cellular components measured by scintillation counting
Assay data:87 Active, 51 Activity ≤ 1 µM, 927 Tested
Binding affinity towards human PGR in an in vitro cell free assay measured by fluorescence polarization method in vitro cell free assay
Assay data:15 Active, 5 Activity ≤ 1 µM, 357 Tested
Antagonist activity at human PGR in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:29 Active, 4 Activity ≤ 1 µM, 850 Tested
Binding affinity towards human OPRK1 in an in vitro assay with cellular components measured by membrane filtration, scintillation proximity assay
Assay data:179 Active, 30 Activity ≤ 1 µM, 1124 Tested
Binding affinity towards human NR3C1 in an in vitro cell free assay measured by filtration, radioactivity method
Assay data:83 Active, 2 Activity ≤ 1 nM, 58 Activity ≤ 1 µM, 1095 Tested
Antagonist activity at human NR3C1 in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:10 Active, 3 Activity ≤ 1 µM, 160 Tested
Binding affinity towards human AR in an in vitro assay with cellular components measured by scintillation counting
Assay data:69 Active, 48 Activity ≤ 1 µM, 927 Tested
Binding affinity towards rat Ar in an in vitro cell free assay measured by fluorescence polarization method
Assay data:45 Active, 19 Activity ≤ 1 µM, 667 Tested
Binding affinity towards human ADORA3 (agonistic activity) in an in vitro assay with cellular components measured by scintillation counting
Assay data:92 Active, 18 Activity ≤ 1 µM, 754 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: KMS28BM_JCRB cell viability assay
Assay data:615 Active, 4 Activity ≤ 1 nM, 321 Activity ≤ 1 µM, 1911 Tested
SummaryPubMed Citation
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: KMS11_JCRBsus cell viability assay
Assay data:722 Active, 10 Activity ≤ 1 nM, 338 Activity ≤ 1 µM, 1911 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: OPM2_DSMZ cell viability assay
Assay data:508 Active, 8 Activity ≤ 1 nM, 210 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: RPMI8226_ATCC cell viability assay
Assay data:685 Active, 11 Activity ≤ 1 nM, 288 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: PCM6_Riken cell viability assay
Assay data:827 Active, 17 Activity ≤ 1 nM, 293 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: PE2_PLB cell viability assay
Assay data:851 Active, 15 Activity ≤ 1 nM, 274 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: UTMC2_PLB cell viability assay
Assay data:584 Active, 49 Activity ≤ 1 nM, 617 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: VP6_DJ cell viability assay
Assay data:933 Active, 17 Activity ≤ 1 nM, 466 Activity ≤ 1 µM, 1912 Tested
Quantitative High-Throughput drug screen in 47 multiple myeloma cell lines against the NCATS MIPE library collection: XG1_PLB cell viability assay
Assay data:892 Active, 13 Activity ≤ 1 nM, 345 Activity ≤ 1 µM, 1912 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on