BioAssays, Active for PubChem Compound (Select 3707) - PubChem BioAssay - NCBI

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Select item 19243951.

Inhibition of recombinant recombinant rat GSK3beta using GS-1 peptide as substrate in presence of [gamma-32P]ATP measured after 30 mins incubation by scintillation counting analysis

Source:: ChEMBL

Protein Target:: Glycogen synthase kinase-3 beta

Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested

AID:: 1924395

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19243942.

Inhibition of recombinant Plasmodium falciparum GSK3 using GS-1 peptide as substrate in presence of [gamma-32P]ATP measured after 30 mins incubation by scintillation counting analysis

Source:: ChEMBL

Assay data:6 Active, 4 Activity ≤ 1 µM, 7 Tested

AID:: 1924394

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953953.

Inhibition of VEGFR (unknown origin)

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895395

Summary Compounds, Active PubMed Citation

Select item 18953944.

Inhibition of FGFR1 (unknown origin)

Source:: ChEMBL

Protein Target:: Fibroblast growth factor receptor 1

Assay data:1 Active, 1 Tested

AID:: 1895394

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 18953785.

Inhibition of FLT3 (unknown origin)

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested

AID:: 1895378

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18953466.

Inhibition of porcine brain GSK-3alpha/beta incubated for 30 mins in presence of [33p]-gamma ATP by scintillation counter analysis

Source:: ChEMBL

Assay data:3 Active, 3 Activity ≤ 1 µM, 5 Tested

AID:: 1895346

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953457.

Inhibition of GST-fused CDK5/p25 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cyclin-dependent kinase 5 activator 1; ...
Total:: 2

Assay data:3 Active, 2 Activity ≤ 1 µM, 5 Tested

AID:: 1895345

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18953218.

Antiproliferative activity against HUVEC cells assessed as cell growth inhibition measured after 3 days by [3H]-thymidine incorporation assay

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895321

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953209.

Antiangiogenic activity in transgenic zebrafish embryo assessed as inhibition of angiogenic vessel growth incubated for 24 hrs by FITC staining based analysis

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895320

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 189531710.

Antiproliferative activity against human MV4-11 cells assessed as cell growth inhibition measured after 72 hrs by tetrazolium staining based WST-8 assay

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895317

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 189531611.

Inhibition of recombinant FLT3 D835Y mutant (unknown origin) in presence of ATP by HTRF assay

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895316

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531512.

Inhibition of recombinant FLT3 (unknown origin) in presence of ATP by HTRF assay

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895315

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531413.

Antiproliferative activity against human OZ [Human cholangiocarcinoma] cells assessed as cell growth inhibition measured upto 72 hrs by CCK-8 assay

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895314

Summary Compounds, Active PubMed Citation

Select item 189531314.

Antiproliferative activity against human HuCCT-1 cells assessed as cell growth inhibition measured upto 72 hrs by CCK-8 assay

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895313

Summary Compounds, Active PubMed Citation

Select item 189531215.

Antiproliferative activity against human NOZ cells assessed as cell growth inhibition measured upto 72 hrs by CCK-8 assay

Source:: ChEMBL

Assay data:1 Active, 1 Tested

AID:: 1895312

Summary Compounds, Active PubMed Citation

Select item 189531116.

Inhibition of SGK (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase Sgk1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895311

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531017.

Inhibition of LCK (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase Lck

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895310

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189530918.

Inhibition of AMPK (unknown origin) in presence of ATP

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895309

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 189530819.

Inhibition of GSK3beta (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Glycogen synthase kinase-3 beta

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895308

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189530720.

Inhibition of GST-fused human CDK2/cyclin A expressed in Escherichia coli using histone H1 as substrate in presence of [33p]-gamma ATP and MgATP

Source:: ChEMBL

Protein Targets:: Cyclin-A2; ...
Total:: 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895307

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Proteins (40)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (151)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (24)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (104)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (125)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (9)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

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BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (88)
BioAssays extracted from the literature
NIH MLP (45)
BioAssays deposited by the NIH Molecular Libraries Program
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BioAssays deposited by other experimentalists

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