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qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT
Assay data:49946 Active, 2 Activity ≤ 1 nM, 3516 Activity ≤ 1 µM, 424035 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT
Assay data:64212 Active, 1 Activity ≤ 1 nM, 3794 Activity ≤ 1 µM, 424003 Tested
Luminescence-based cell-based primary high throughput screening assay to identify activators of the DAF-12 from the parasite H. contortus (hcDAF-12)
Assay data:5354 Active, 370276 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS of Nrf2 Activators
Assay data:1243 Active, 151 Activity ≤ 1 µM, 407090 Tested
qHTS profiling assay for firefly luciferase inhibitor/activator using purifed enzyme and Km concentrations of substrates (counterscreen for miR-21 project)
Assay data:25159 Active, 3019 Activity ≤ 1 µM, 364105 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Screen for inhibitors of the SWI/SNF chromatin remodeling complex (esBAF) in mouse embryonic stem cells with Luciferase reporter assay Measured in Cell-Based System Using Plate Reader - 2141-01_Inhibitor_SinglePoint_HTS_Activity
Assay data:7048 Active, 347670 Tested
HTS Assay for Compounds that Act as Agonists of the Vanilloid Receptor 1
Assay data:617 Active, 316974 Tested
qHTS screen for small molecules that inhibit ELG1-dependent DNA repair in human embryonic kidney (HEK293T) cells expressing luciferase-tagged ELG1
Assay data:7656 Active, 3127 Activity ≤ 1 µM, 330279 Tested
Dose Response for ABC transporter inhibitors: specifically ABCG2 screen, ABCB1 counter-screen. Follow-up assay.
Assay data:75 Active, 12 Activity ≤ 1 µM, 89 Tested
qHTS Assay for Antagonists of the Neuropeptide S Receptor: cAMP Signal Transduction
Assay data:2314 Active, 1 Activity ≤ 1 nM, 558 Activity ≤ 1 µM, 221370 Tested
A qHTS for Small Molecule Inhibitors of Shiga Toxin
Assay data:26913 Active, 293642 Tested
Cycloheximide Counterscreen for Small Molecule Inhibitors of Shiga Toxin
Assay data:37055 Active, 296456 Tested
Single point confirmation screening for ABC transporter inhibitors: specifically ABCG2 screen, ABCB1 counter-screen
Assay data:16 Active, 273 Tested
Single point confirmation for ABC transporter inhibitors: specifically ABCB1 screen, ABCG2 counter-screen
Assay data:18 Active, 273 Tested
High-throughput multiplex screening for ABC transporter inhibitors: specifically ABCB1 screen, ABCG2 counter-screen
Assay data:130 Active, 193717 Tested
High-throughput multiplex screening for ABC transporter inhibitors: specifically ABCG2 screen, ABCB1 counter-screen
Assay data:200 Active, 194480 Tested
Primary cell-based high throughput screening assay to measure STAT3 activation
Assay data:1773 Active, 194698 Tested
Chemo Reversal assay in ABCB1-expressing cells for one set of SAR compounds
Assay data:1 Active, 15 Tested
Chemo Reversal assay in ABCG2-expressing cells for one set of SAR compounds
Assay data:5 Active, 15 Tested
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