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Experimentally measured binding affinity data (IC50) for protein-ligand complexes derived from PDB
Assay data:4302 Active, 250 Activity ≤ 1 nM, 2931 Activity ≤ 1 µM, 4302 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition of human recombinant APP in CHO cells assessed as decrease in beta amyloid protein level by ELISA
Assay data:10 Active, 2 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of BACE2 by FRET assay
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
Inhibition of human recombinant BACE1 expressed CHO cells by FRET assay
Assay data:27 Active, 17 Activity ≤ 1 µM, 27 Tested
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