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Compound was evaluated for the inhibition of human recombinant SAMHD1 at 5uM in a enzyme-coupled malachite green assay
Assay data:17606 Tested
SummaryPubMed CitationRelated BioAssays by Target
Permeability of the compound across blood brain barrier at pH 7.4 at 50 uM incubated for 4 hrs by PAMPA assay
Assay data:2 Tested
SummaryPubMed Citation
Effective permeability of compound by PAMPA-BBB assay
Assay data:6 Tested
Effective permeability of compound at 25 ug/ml incubated for 18 hrs by PAMPA-BBB assay
Assay data:19 Tested
Permeability of the compound incubated for 18 hrs by PAMPA-BBB assay
Assay data:16 Tested
Effective permeability of compound by PAMPA-BBA method
Assay data:5 Tested
Solubility of compound in 1:99 DMSO/PBS incubated for 4 hrs
Assay data:2 Active, 1 Activity ≤ 1 µM, 13 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
HIV Enzyme Data
Assay data:46810 Tested
Summary
HIV Cellular Data
Assay data:126857 Tested
p53 small molecule agonists, cell-based qHTS assay with human liver microsomes: Summary
Assay data:70 Active, 12 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
p53 small molecule agonists, cell-based qHTS assay: Summary
Assay data:212 Active, 41 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
p53 small molecule agonists, cell-based qHTS assay with rat liver microsomes: Summary
Assay data:103 Active, 14 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay
Assay data:87 Active, 5 Activity ≤ 1 nM, 180 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay: qHTS cell viability counter screen
Assay data:213 Active, 2 Activity ≤ 1 nM, 241 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay with rat liver microsomes: qHTS cell viability counter screen
Assay data:214 Active, 153 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay with human liver microsomes: qHTS cell viability counter screen
Assay data:300 Active, 138 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay with rat liver microsomes
Assay data:27 Active, 44 Activity ≤ 1 µM, 9667 Tested
p53 small molecule agonists, cell-based qHTS assay with human liver microsomes
Assay data:43 Active, 55 Activity ≤ 1 µM, 9667 Tested
Primary qHTS assay for Inhibitors of ovarian cancer metastasis using an organotypic tumor microenvironment (TME) model.
Assay data:60 Active, 47 Activity ≤ 1 µM, 45897 Tested
HTS to identify compounds that affect the blood-brain barrier permeability in vitro
Assay data:419 Active, 1260 Tested
SummaryCompounds, Active
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