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Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in HEK293 cells by scintillation counting analysis
Assay data:1 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]-Diprenorphine from human KOP receptor expressed in HEK293 cells by scintillation counting method
Assay data:1 Active, 3 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Displacement of [3H]-Diprenorphine from human DOP receptor expressed in HEK293 cells by scintillation counting method
Assay data:1 Active, 1 Activity ≤ 1 µM, 11 Tested
Displacement of [3H]-Diprenorphine from human MOP receptor expressed in HEK293 cells by scintillation counting method
Assay data:1 Active, 2 Activity ≤ 1 µM, 11 Tested
Displacement of [125I]-43RFa from human QRFP receptor expressed in CHO cells by TopCount scintillation counting method
Displacement of [125I]-Kp-10 from human Kiss1 receptor by TopCount scintillation counting method
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 11 Tested
Displacement of [3H]-PrRP-20 from human PrRP receptor expressed in CHO cells by TopCount scintillation counting method
Agonist activity at human mu opioid receptor expressed in CHO cells assessed as dynamic mass redistribution by DMR assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
Agonist activity at human NOP receptor expressed in CHO cells assessed as dynamic mass redistribution by DMR assay relative to control
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at human NOP receptor expressed in CHO cells assessed as dynamic mass redistribution by DMR assay
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 3 Tested
Concentration ratio of human mu opioid receptor expressed in CHO cells to human NOP receptor expressed in CHO cells
Assay data:3 Tested
SummaryPubMed Citation
Enzymatic assay of human HDAC6 with custom peptide substrate
Assay data:5603 Tested
SummaryRelated BioAssays by Target
Enzymatic assay of human HDAC6 with commercial peptide substrate
Antiviral activity determined as inhibition of SARS-CoV-2 induced cytotoxicity of VERO-6 cells at 10 uM after 48 hours exposure to 0.01 MOI SARS CoV-2 virus by high content imaging
Assay data:7212 Tested
Summary
SARS-CoV-2 3CL-Pro protease inhibition percentage at 20 M by FRET kind of response from peptide substrate
Antiviral activity determined as inhibition of SARS-CoV-2 induced cytotoxicity of Caco-2 cells at 10 uM after 48 hours by high content imaging
Assay data:5612 Tested
Mouse NOP receptor (Opioid receptors)
Assay data:5 Active, 5 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Human NOP receptor (Opioid receptors)
Assay data:30 Active, 30 Tested
Agonist activity at human nociceptin receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP production preincubated for 15 mins followed by forskolin addition measured for 90 mins by luciferase reporter gene assay
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]nociceptin from human recombinant Nociceptin receptor expressed in HEK293 cells
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
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