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Binding affinity to recombinant human adenosine A2B receptor expressed in CHO cell membranes at 100 nM after 15 mins in presence of DPCPX by confocal microscopic method
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to recombinant human adenosine A2B receptor expressed in CHO cell membranes at 100 nM after 15 mins in presence of PSB-603 by confocal microscopic method
Binding affinity to wild type CHO cell membranes at 100 nM after 15 mins by confocal microscopic method
SummaryPubMed Citation
Binding affinity to recombinant human adenosine A2B receptor expressed in CHO cell membranes at 100 nM after 15 mins by confocal microscopic method
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antagonist activity at recombinant human adenosine A2B receptor expressed in CHO cell membranes assessed as inhibition of NECA-induced cAMP accumulation preincubated for 1 hr followed by NECA induction measured after 5 mins in presence of [3H]cAMP and bovine cAMP-binding protein by liquid scintillation counting method
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Selectivity ratio of Ki for recombinant human adenosine A3 receptor expressed in CHO cell membranes to Ki for recombinant rat adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A3 receptor expressed in CHO cell membranes to Ki for recombinant mouse adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A1 receptor expressed in CHO cell membranes to Ki for recombinant rat adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A1 receptor expressed in CHO cell membranes to Ki for recombinant mouse adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A1 receptor expressed in CHO cell membranes to Ki for recombinant human adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A3 receptor expressed in CHO cell membranes to Ki for recombinant human adenosine A2B receptor expressed in CHO cell membranes
Assay data:2 Tested
Selectivity ratio of Ki for adenosine A2A receptor in rat brain striatal membranes to Ki for recombinant rat adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A2A receptor expressed in HEK cell membranes to Ki for recombinant rat adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A2A receptor expressed in HEK cell membranes to Ki for recombinant mouse adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for adenosine A2A receptor in rat brain striatal membranes to Ki for recombinant mouse adenosine A2B receptor expressed in CHO cell membranes
Selectivity ratio of Ki for recombinant human adenosine A2A receptor expressed in HEK cell membranes to Ki for recombinant human adenosine A2B receptor expressed in CHO cell membranes
Assay data:3 Tested
Selectivity ratio of Ki for adenosine A2A receptor in rat brain striatal membranes to Ki for recombinant human adenosine A2B receptor expressed in CHO cell membranes
Assay data:9 Tested
Displacement of [3H]PSB-11 from recombinant human adenosine A3 receptor expressed in CHO cell membranes after 45 mins by liquid scintillation counting method
Assay data:6 Active, 3 Activity ≤ 1 µM, 9 Tested
Displacement of [3H]PSB-603 from recombinant mouse adenosine A2B receptor expressed in CHO cell membranes after 75 mins by liquid scintillation counting method
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Displacement of [3H]PSB-603 from recombinant rat adenosine A2B receptor expressed in CHO cell membranes after 75 mins by liquid scintillation counting method
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 2 Tested
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