BioAssays for PubChem Compound (Select 101375) - PubChem BioAssay - NCBI

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Items: 10

Select item 17982241.

Enzyme Inhibition Assay from Article 10.1021/jm049011j: "Identification and characterization of novel benzil (diphenylethane-1,2-dione) analogues as inhibitors of mammalian carboxylesterases."

Source:: BindingDB

Protein Targets:: Acetylcholinesterase; ...
Total:: 5

Assay data:36 Active, 30 Activity ≤ 1 µM, 60 Tested

AID:: 1798224

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 4122362.

Lipophilicity, log P of the compound

Source:: ChEMBL

Assay data:41 Tested

AID:: 412236

Summary PubMed Citation

Select item 4122293.

Inhibition of rabbit carboxylesterase

Source:: ChEMBL

Assay data:32 Active, 30 Activity ≤ 1 µM, 32 Tested

AID:: 412229

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 4122284.

Inhibition of human carboxylesterase 1

Source:: ChEMBL

Protein Target:: Liver carboxylesterase 1

Assay data:28 Active, 22 Activity ≤ 1 µM, 30 Tested

AID:: 412228

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 4122275.

Inhibition of human intestinal carboxylesterase

Source:: ChEMBL

Assay data:31 Active, 28 Activity ≤ 1 µM, 31 Tested

AID:: 412227

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 2392726.

Inhibition constant against human intestinal carboxylesterase 2 (hiCE) using nitrophenyl acetate (o-NPA) as substrate

Source:: ChEMBL

Protein Target:: Cocaine esterase

Assay data:31 Active, 26 Activity ≤ 1 µM, 61 Tested

AID:: 239272

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2391977.

Inhibition constant against human liver carboxylesterase 1 (hCE1) using nitrophenyl acetate (o-NPA) as substrate

Source:: ChEMBL

Protein Target:: Liver carboxylesterase 1

Assay data:26 Active, 18 Activity ≤ 1 µM, 61 Tested

AID:: 239197

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2391678.

Inhibition constant against rabbit liver carboxylesterase (rCE) using nitrophenyl acetate (o-NPA) as substrate

Source:: ChEMBL

Protein Target:: Liver carboxylesterase 1

Assay data:32 Active, 28 Activity ≤ 1 µM, 61 Tested

AID:: 239167

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2391669.

Inhibition constant against human Butyrylcholinesterase (hBuChE) using butyrylthiocholine (BuTCh) as substrate

Source:: ChEMBL

Protein Target:: Cholinesterase

Assay data:3 Active, 1 Activity ≤ 1 µM, 61 Tested

AID:: 239166

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 23912210.

Inhibition constant against human Acetylcholinesterase (hAcChE) using acetylthiocholine (AcTCh) as substrate

Source:: ChEMBL

Protein Target:: Acetylcholinesterase

Assay data:3 Active, 2 Activity ≤ 1 µM, 61 Tested

AID:: 239122

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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BioActivity

Active Compounds (9)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 µM (9)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (9)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (10)
BioAssays extracted from the literature

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