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Selectivity interaction (Enzyme panel (Eurofins-Cerep)) EUB0000262b UTS2R
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (CEREP panel (Eurofins, binding assay)) EUB0000262b UTS2R
UT (h) Eurofins-Cerep binding assay
Assay data:2 Tested
PRESTO-Tango GPCRome screening (UTS2R)
UROTENSIN_II Eurofins-Panlabs selectivity data (BI)
UT1/H AG Cerep selectivity data (BI)
UT (h) CEREP ligand profiling
UROTENSIN_II Eurofins SafetyScreen44 (BI)
Agonist activity at human U-IIR expressed in HEK293-A cells at >500 nM by Fluo4-AM dye based intracellular calcium mobilization assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at human U-IIR expressed in HEK293-A cells at 500 nM by Fluo4-AM dye based intracellular calcium mobilization assay relative to control
Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand binding assay
Assay data:13 Active, 1 Activity ≤ 1 nM, 7 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at human U-IIR expressed in HEK293-A cells assessed as delta F/F0 ratio by Fluo4-AM dye based intracellular calcium mobilization assay
Assay data:32 Tested
Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assay
Assay data:32 Active, 2 Activity ≤ 1 nM, 32 Activity ≤ 1 µM, 34 Tested
Antagonist activity at human UT receptor expressed in HEK293 cells using Na [125I] incubated for 2 hrs by gamma counting method
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
Agonist activity at urotensin 2 receptor (unknown origin) expressed in HEK293 cells co-expressing Gq-polycistronic BRET biosensor assessed as induction of Gq activation measured for 5 mins by luminescence detection based BRET assay relative to URP
Assay data:11 Tested
Agonist activity at urotensin 2 receptor (unknown origin) expressed in HEK293 cells co-expressing Gq-polycistronic BRET biosensor assessed as induction of Gq activation measured for 5 mins by luminescence detection based BRET assay
Assay data:12 Active, 12 Activity ≤ 1 µM, 12 Tested
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