Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 19592201.

Inhibition of BCRP (unknown origin) expressed in dog MDCK-II cells assessed as maximum inhibition using pheophorbide A as substrate preincubated for 20 mins followed by substrate addition and measured after 120 mins by flow cytometry analysis relative to control

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Tested

AID:: 1959220

Summary PubMed Citation Related BioAssays by Target

Select item 19592152.

Inhibition of BCRP (unknown origin) expressed in dog MDCK-II cells at 10 uM using pheophorbide A as substrate preincubated for 20 mins followed by substrate addition and measured after 120 mins by flow cytometry analysis relative to control

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:34 Tested

AID:: 1959215

Summary PubMed Citation Related BioAssays by Target

Select item 19592123.

Inhibition of BCRP (unknown origin) expressed in dog MDCK-II cells using pheophorbide A as substrate preincubated for 20 mins followed by substrate addition and measured after 120 mins by flow cytometry analysis

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:13 Active, 1 Activity ≤ 1 µM, 23 Tested

AID:: 1959212

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19592094.

Inhibition of BCRP (unknown origin)

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 2 Tested

AID:: 1959209

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 19592085.

Inhibition of BCRP (unknown origin) by Hoechst 33342 staining based assay

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Tested

AID:: 1959208

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 19592066.

Inhibition of BCRP (unknown origin) expressed in MDCK cells assessed as increase in Hoechst 33342 accumulation incubated for 60 mins by Hoechst 33342 dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1959206

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19592047.

Inhibition of BCRP (unknown origin) expressed in MDCK cells assessed as increase in Hoechst 33342 accumulation incubated for 30 mins by Hoechst 33342 dye based fluorescence assay

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Tested

AID:: 1959204

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 19481068.

Binding affinity to ABCG2 in vincristine resistant human Eca-109 cells assessed as stabilization of protein at 100 uM incubated for 30 mins by thermal shift assay

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Tested

AID:: 1948106

Summary PubMed Citation Related BioAssays by Target

Select item 19479649.

Substrate activity at human BCRP in dog MDCKII-MDR1 cells using 14C-labeled ligand

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Tested

AID:: 1947964

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 194219710.

Inhibition of ABCG2 (unknown origin)

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested

AID:: 1942197

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 192300511.

Substrate activity at mouse BCRP assessed as apparent permeability at 1 uM

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:9 Tested

AID:: 1923005

Summary PubMed Citation Related BioAssays by Target

Select item 192300412.

Substrate activity at mouse BCRP assessed as efflux ratio at 1 uM

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:9 Tested

AID:: 1923004

Summary PubMed Citation Related BioAssays by Target

Select item 191698213.

Inhibition of ABCG2 (unknown origin) in Sf9 membrane vesicles using [3H] methotrexate as substrate

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:2 Tested

AID:: 1916982

Summary PubMed Citation Related BioAssays by Target

Select item 191697914.

Inhibition of ABCG2 (unknown origin) overexpressing in dog MDCK-II-BCRP cells

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1916979

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191697815.

Inhibition of ABCG2 (unknown origin) overexpressing in dog MDCK-II-BCRP cells measured after 30 mins by flow cytometric analysis

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Tested

AID:: 1916978

Summary PubMed Citation Related BioAssays by Target

Select item 191697716.

Inhibition of ABCG2 in HEK293 cells

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1916977

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191697617.

Inhibition of wildtype ABCG2 (unknown origin) transfected in HEK293 cells measured after 30 mins by flow cytometric anlaysis

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1916976

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191697518.

Inhibition of ABCG2 (unknown origin)

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1916975

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 190412419.

Inhibition of BCRP (unknown origin)

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1904124

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 190218620.

Inhibition of human ABCG2 in human R5 cells assessed as inhibition of mitoxantrone efflux measured by flow cytometric analysis

Source:: ChEMBL

Protein Target:: Broad substrate specificity ATP-binding cassette transporter ABCG2

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1902186

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Target

Proteins (11)
BioAssays with protein sequences specified as targets

BioActivity

Chemical Probes (1)
BioAssays with compounds reported as validated chemical probes

Active Compounds (377)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (3)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (192)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (279)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (3)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose

Assay Project (8)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (771)
BioAssays extracted from the literature
NIH MLP (8)
BioAssays deposited by the NIH Molecular Libraries Program
Other (127)
BioAssays deposited by other experimentalists

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