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In Vitro Enzyme IC50 Assay from US Patent US20240207292: "BORONIC ACID COMPOUNDS, COMPOSITIONS AND METHODS"
Assay data:93 Active, 7 Activity ≤ 1 nM, 93 Activity ≤ 1 µM, 93 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
DPP4 activity assay from US Patent US20240115577: "SMALL MOLECULE REGULATORS OF ALVEOLAR TYPE 2 CELL PROLIFERATION FOR THE TREATMENT OF PULMONARY DISEASES"
Assay data:25 Active, 9 Activity ≤ 1 nM, 25 Activity ≤ 1 µM, 25 Tested
Inhibition of mouse DPP4
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human recombinant DPP-4 at 25 uM using Gly-Pro-Aminomethylcoumarin as substrate by Spectra max fluorometer analysis relative to control
Inhibition of human recombinant DPP-4 at 10 uM using Gly-Pro-Aminomethylcoumarin as substrate by Spectra max fluorometer analysis relative to control
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human recombinant DPP-4 at 100 uM using Gly-Pro-Aminomethylcoumarin as substrate by Spectra max fluorometer analysis relative to control
Assay data:6 Tested
Inhibition of human recombinant DPP-4 at 10 uM relative to control
Binding affinity to DPP-4 (unknown origin) assessed as inhibition constant
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human recombinant DPP-4 using H-Gly-Pro-aminomethylcoumarin as substrate at 100 uM relative to control
Assay data:2 Tested
Inhibition of human recombinant DPP-4 using H-Gly-Pro-aminomethylcoumarin as substrate
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of DPP-4 (unknown origin) at 100 uM relative to control
Assay data:4 Tested
Inhibition of DPP-4 (unknown origin) using (H-Gly-Pro-AMC) as substrate
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of human recombinant DPP-4
Assay data:9 Active, 8 Activity ≤ 1 µM, 9 Tested
Inhibition of human recombinant DPP-4 using (H-Gly-Pro-AMC as substrate
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
Inhibition of human DPP-4 expressed in human Caco-2 cells using H-Gly-Pro-AMC as substrate measured for 30 mins by microplate reader analysis
Assay data:13 Active, 11 Activity ≤ 1 nM, 13 Activity ≤ 1 µM, 13 Tested
Inhibition of DPP-4 (unknown origin) relative to control
Assay data:7 Tested
Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate incubated for 30 mins by spectroscopic analysis
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of DPP-4 (unknown origin)
Assay data:83 Active, 14 Activity ≤ 1 nM, 80 Activity ≤ 1 µM, 87 Tested
Inhibition of recombinant human dipeptidyl peptidase 4 using Gly-Pro-AMC as substrate
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of DPP4 (unknown origin)
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