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Determination of FXIIa Inhibition from US Patent US20240059691: "ENZYME INHIBITORS"
Assay data:275 Active, 166 Activity ≤ 1 µM, 340 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Cross screening panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Safety47 Scan (DiscoverX - Eurofins)
Cholinesterase, Acetyl, ACES Eurofins Panlabs panel
Compound was evaluated for inhibition of human ACHE in an vitro cell free assay measured by absorbance method
Assay data:10 Active, 5 Activity ≤ 1 µM, 73 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Assay data:31 Active, 15 Activity ≤ 1 µM, 927 Tested
Inhibition of AChE (unknown origin) upto 10000 nM
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of AChE (unknown origin) by UV spectrophotometric analysis
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
Inhibition of AChE (unknown origin)
Assay data:13 Active, 13 Activity ≤ 1 µM, 14 Tested
Inhibition of human AchE
Inhibition of BChE (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Inhibition of human AChE using acetylthiocholine iodide as substrate preincubated with enzyme for 20 mins followed by substrate addition and measured for 5 mins by Ellman's spectrophotometric method
Assay data:19 Active, 5 Activity ≤ 1 µM, 20 Tested
Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated with enzyme for 20 mins followed by substrate addition and measured for 5 mins by Ellman's spectrophotometric method
Assay data:6 Active, 6 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human BChE using butyrylthiocholine iodide as substrate at 10 uM preincubated with enzyme for 20 mins followed by substrate addition and measured for 5 mins by Ellman's spectrophotometric method
Assay data:6 Tested
Competitive inhibition of human AChE using acetylthiocholine iodide as substrate preincubated with enzyme for 20 mins followed by varing concentrations of substrate addition and measured for 5 mins by Lineweaver-Burk plot analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate at 50 to 100 uM preincubated for 20 mins followed by substrate addition and measured after 20 mins by Ellman's method
Assay data:24 Tested
Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated with compounds for 20 mins followed by substrate addition and measured after 20 mins by Ellman's method relative to control
Assay data:4 Active, 2 Activity ≤ 1 µM, 6 Tested
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