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Agonist activity at human TRPM4 expressed in CHO-K1 cells assessed as increase in relative fluorescence unit by measuring membrane potential by FLIPR assay
Assay data:5 Active, 1 Activity ≤ 1 µM, 9 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at human TRPM4 at <= 30 uM
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assay
Assay data:1 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of TRPM4 channel (unknown origin)
Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx up to 100 uM after 45 mins by ANG2 dye-based fluorescence assay
Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx at 10 uM after 45 mins by ANG2 dye-based fluorescence assay relative to control
Inhibition of TRPM4 (unknown origin)
Inhibition of Flag-tagged TRPM4 (unknown origin) expressed in HEK293 cells assessed as reduction in intracellular Na+ influx after 45 mins by ANG2 dye-based fluorescence assay
Assay data:9 Active, 1 Activity ≤ 1 µM, 9 Tested
Inhibition of TRPM4 in human Jurkat T cells assessed as reduction in intracellular calcium flux at 500 nM within 60 mins by whole cell patch clamp electrophysiology method
Mouse TRPM4 (Transient Receptor Potential channels)
Assay data:4 Active, 4 Tested
Human TRPM4 (Transient Receptor Potential channels)
Assay data:12 Active, 12 Tested
Inhibition of TRPM4 (unknown origin) expressed in HEK293 cells assessed as effect on agonist-induced Ca2+ changes
SummaryRelated BioAssays by Target
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