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Inhibition of rat liver SULT1A1-mediated oestradiol sulfonation incubated for 20 mins
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Amoxapine and Protriptyline Inhibition Assay from Article 10.1074/jbc.M113.510974: "High accuracy in silico sulfotransferase models."
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax/Km ratio incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis
Assay data:25 Tested
SummaryRelated BioAssays by Target
Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Vmax incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis
Substrate activity at SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells assessed as substrate Km incubated for 15 mins using [35S-]PAPS as sulfate donor by TLC analysis
Assay data:14 Active, 9 Activity ≤ 1 µM, 25 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of SULT1A1 (unknown origin) expressed in baculovirus infected Sf9 cells incubated for 15 mins using para-nitrophenol as substrate by TLC analysis
Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation measured per mg of protein after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS
Assay data:1 Tested
Activity of human SULT1A1 expressed in escherichia coli assessed as enzyme-mediated 4-(4-chloro-1-(4-(2-(dimethylamino)ethoxy)phenyl)-2-phenylbut-1-enyl)phenyl hydrogen sulfate formation after 15 mins by Michaelis-Menten equation in presence of 20 uM PAPS
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of SULT1A1 in human MCF7 cells assessed as 17beta-estradiol sulfation
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of human SULT1A1 expressed in Escherichia coli assessed as beta-naphthol sulfation at 100 nM by Michaelis-Menten equation analysis
Inhibition of human SULT1A1 expressed in Escherichia coli assessed as p-nitrophenol sulfation at 100 nM by Michaelis-Menten equation analysis
Inhibition of human SULT1A1 expressed in Escherichia coli assessed as 17beta-estradiol sulfation at 100 nM by Michaelis-Menten equation analysis
Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence in presence of 3',5'-phosphoadenosine
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence
Activity of human SULT1A1 expressed in Escherichia coli at 6 uM by Michaelis-Menten equation analysis in presence of PAPS
Activity of human SULT1A1 expressed in Escherichia coli at 6 uM by Michaelis-Menten equation analysis
Activity of human SULT1A1 expressed in Escherichia coli at 20 uM by Michaelis-Menten equation analysis in presence of PAPS
Activity of human SULT1A1 expressed in Escherichia coli at 20 uM by Michaelis-Menten equation analysis
Activity of human SULT1A3 assessed as compound formation treated with 2 and 20 uM brivanib for 30 mins by LC/MS analysis in presence of PAPS
Activity of human SULT1A1 assessed as compound formation treated with 2 and 20 uM brivanib for 30 mins by LC/MS analysis in presence of PAPS
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