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assay on hold
Summary
Inhibition of CDK2/cyclin A (unknown origin) at 10 uM by biochemical hotspot kinase assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of ERK2 (unknown origin) at 10 uM by biochemical hotspot kinase assay relative to control
Inhibition of c-Src (unknown origin) at 10 uM by biochemical hotspot kinase assay
Inhibition of FGFR2 (unknown origin) at 10 uM by biochemical hotspot kinase assay
Inhibition of GST-tagged human CDK2/Cyclin A2 expressed in baculovirus infected Sf9 cells using 5-FAM-QSPKKG-CONH2 as substrate at 10 uM incubated for 60 mins in presence of ATP relative to control
Inhibition of GST-tagged human CDK2/Cyclin A2 expressed in baculovirus infected Sf9 cells using 5-FAM-QSPKKG-CONH2 as substrate incubated for 60 mins in presence of ATP
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of STAT5 phosphorylation at Tyr694 residue in human MV4-11 cells harboring FLT3-ITD mutant incubated for 4 hrs by Western blot analysis
Inhibition of STAT5 phosphorylation at Tyr694 residue in human MOLM-14 cells harboring FLT3-ITD mutant incubated for 4 hrs by Western blot analysis
Inhibition of STAT5 phosphorylation at Tyr694 residue in human MOLM-13 cells harboring FLT3-ITD mutant incubated for 4 hrs by Western blot analysis
Binding affinity to Estrogen receptor alpha (unknown origin) at 1 uM by displacement assay relative to control
Inhibition of FGFR (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of CDK2/cyclin E1 (unknown origin) expressed in Sf9 cells
Assay data:2 Active, 9 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of BMI1 (unknown origin) by ELISA assay
Assay data:25 Active, 25 Activity ≤ 1 nM, 25 Activity ≤ 1 µM, 25 Tested
Inhibition of CDK2/cyclin E (unknown origin)
Assay data:5 Active, 10 Tested
Inhibition of Src (unknown origin) at 1 uM relative to control
Assay data:3 Tested
Inhibition of CDK2/cyclin A (unknown origin) at 1 uM relative to control
Binding affinity to human partial length TRIM24 (P790 to P977 residues) expressed in bacterial expression system by BROMOscan assay
Assay data:4 Tested
Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assay
Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assay
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