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Binding affinity towards human SLC29A1 in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:20 Active, 4 Activity ≤ 1 µM, 1115 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human Nav1.6 alpha subunit expressed in HEK293 cells co-expressing beta1 subunit at -35 mV holding potential by PatchXpress automated voltage clamp electrophysiology technique
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of calmodulin (unknown origin)
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of PTP1B (unknown origin) by DAS-ELISA
Assay data:7 Active, 6 Activity ≤ 1 µM, 7 Tested
Inhibition of PTP1B (unknown origin) at 10 micromol/L by DAS-ELISA
Assay data:29 Tested
Inhibition of PTP1B (unknown origin) using pNPP as substrate preincubated for 10 mins followed by substrate addition and measured every 30 sec for 10 mins by microplate photometer analysis
Assay data:5 Tested
Antagonist activity at SMO D473H mutant (unknown origin) expressed in mouse TM3 cells coexpressing Gli-luc reporter gene assessed as inhibition of Hh-Ag1.5 induced Gli luciferase activity incubated for 48 hrs by luminescence assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of human PRMT4 by fluorescence-based SAHH-coupled assay
Inhibition of ACAT in human THP-1
Assay data:4 Active, 5 Activity ≤ 1 µM, 5 Tested
Inhibition of human recombinant GST-tagged PTP1B (1 to 321 residues) expressed in Escherichia coli using pNPP as substrate preincubated for 10 mins followed by substrate addition and measured after 30 mins by microplate reader assay
Assay data:1 Tested
Inhibition of human recombinant PTP1B using pNPP as substrate incubated for 40 min
Inhibition of human PTP1B using pNPP as substrate incubated for 30 min by UV-Visible spectrophotometer assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of PTP1B (unknown origin) using DiFMUP as substrate incubated for 30 min by fluorescence based microplate reader assay
Inhibition of human PTP1B using pNPP as substrate incubated for 30 min by microplate reader assay
Inhibition of human recombinant GST-tagged PTP1B (1 to 321 residues) expressed in Escherichia coli using pNPP as substrate by spectrophotometer assay
Inhibition of PTP1B (unknown origin) using pNPP as substrate
Inhibition of human PTP1B (1 to 411 residues) expressed in Escherichia coli BL21 (DE3) using GNGDpYMPMSPKS as phosphopeptide substrate incubated for 30 mins by malachite green reagent assay
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Inhibition of human recombinant PTP1B expressed in Escherichia coli BL21 (DE3) using pNPP as substrate by high-throughput screening assay
Inhibition of human PTP1B (1 to 298 residues) expressed in Escherichia coli using FDP as substrate by microplate reader
Inhibition of human PTP1B expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant using pNPP as substrate incubated for 15 min by Michaelis-Menten analysis
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