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RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Inhibition of 20S immunoproteasome beta 1 in human Raji cell lysates after 1 hr by competitive ABPP assay
Assay data:17 Tested
SummaryPubMed CitationRelated BioAssays by Target
Potency index, ratio of ixazomib IC50 to compound IC50 for inhibition of human 20S proteasome using Suc-LLVY-AMC as substrate measured every 5 mins for 120 mins by fluorescence based assay
Assay data:2 Tested
Inhibition of 20S proteasome in human BE(2)-C cells at 2xIC50 using LLVY-R110 peptide as substrate measured up to 36 hrs by fluorescence based assay
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of 20S proteasome in human HeLa cells at 2xIC50 using LLVY-R110 peptide as substrate measured up to 36 hrs by fluorescence based assay
Inhibition of human 20S proteasome using Suc-LLVY-AMC as substrate measured every 5 mins for 120 mins by fluorescence based assay
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human immunoproteasome beta 1i subunit using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay
Assay data:10 Tested
Inhibition of human immunoproteasome beta 1i subunit at 10 uM using Ac-PAL-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay
Inhibition of human 26S proteasome using suc-LLVY-AMC as substrate up to 40 mins by fluorescence assay
Inhibition of 20s immunoproteasome LMP2 in human erythrocytes using Ac-Pro-Ala-Leu-MCA as substrate preincubated for 10 mins followed by substrate addition and measured after 6 hrs by fluorescence assay
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Inhibition of 20S immunoproteasome beta 1 in human RPMI8226 cell lysates after 1 hr by coomassie brilliant blue staining-based fluorescence assay
Assay data:9 Tested
Inhibition of LMP2 in human MOLT4 cell lysate after 1 hr by ELISA
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Inhibition of human 20S immunoproteasome beta-1 at 50 uM using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assay relative to control
Assay data:31 Tested
Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assay
Assay data:10 Active, 1 Activity ≤ 1 µM, 24 Tested
Inhibition of 20S proteasome activity in human ANBL-6 cells
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced TNF-alpha response in human macrophages_Primary screen TNF readout
Assay data:2853 Active, 18113 Tested
SummaryRelated BioAssays by Same Project
Inhibition of proteasome subunit beta-1i in human RPMI8226 cells using BODIPY-NC001 by fluorescent densitometry
Assay data:7 Active, 4 Activity ≤ 1 µM, 10 Tested
Inhibition of proteasome subunit beta-1i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry
Assay data:17 Active, 15 Activity ≤ 1 µM, 21 Tested
A screen to identify synthetic lethal interactions with E-cadherin in an MCF10A isogenic cell line
Assay data:2442 Active, 18052 Tested
SummaryPubMed Citation
A screen to identify genes that regulate lymphatic endothelial cell migration - Primary Screen
Assay data:1034 Active, 18120 Tested
SummaryRelated BioAssays by Depositor
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