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Displacement of [3H]-iloprost from recombinant rat IP receptor expressed in CHO-K1 cell membranes incubated for 1 hr by top count scintillation counting method
Assay data:3 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at recombinant rat IP receptor expressed in CHO-K1 cells assessed as increase in intracellular cAMP level after 1 hr incubation by HTRF method
Assay data:20 Active, 1 Activity ≤ 1 nM, 15 Activity ≤ 1 µM, 23 Tested
Intrinsic activity at recombinant rat IP receptor expressed in CHO-K1 cells assessed as increase in intracellular cAMP level at 10 uM after 1 hr incubation by HTRF method relative to iloprost
Assay data:20 Tested
SummaryPubMed CitationRelated BioAssays by Target
Rat IP receptor (Prostanoid receptors)
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Intrinsic activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay relative to 1 uM iloprost
Assay data:32 Tested
Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay
Assay data:28 Active, 25 Activity ≤ 1 µM, 32 Tested
Inhibition of rat I2 receptor at 1 uM
Assay data:1 Tested
Agonist activity at rat PGI2 receptor assessed as inhibition of ADP-induced platelet aggregation
Assay data:2 Active, 1 Activity ≤ 1 µM, 9 Tested
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