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pA2 value against Glucagon Receptor; Not determined
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Compound was evaluated for its ability to displace radiolabeled glucagon (inactive up to 100 uM)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Compound was evaluated for its ability to displace radiolabeled glucagon
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagon
Assay data:13 Active, 12 Activity ≤ 1 µM, 13 Tested
Binding affinity towards rat Glucagon Receptor
Relative binding affinity for rat glucagon receptor compared to glucagon
Assay data:2 Tested
In vitro receptor binding affinity using rat liver plasma membrane bioassay; inactive
Assay data:4 Tested
Assay data:5 Tested
In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Glucagon receptor binding measured as percentage stimulation
Assay data:15 Tested
pA2 value against Glucagon Receptor
pA2 value towards glucagon receptor relative to glucagon was calculated
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
In vitro inhibitory activity against rat glucagon receptor using [127I]-labeled glucagon
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Assay data:11 Active, 11 Activity ≤ 1 µM, 11 Tested
Relative binding by measuring competition for glucagon receptor between [125]glucagon and the compound.
Assay data:29 Tested
Relative binding was evaluated by measuring competition for glucagon receptor between [1-6]glucagon and the compound.
Relative binding potency as ratio of IC50 relative to glucagon binding
Assay data:9 Tested
inhibition of [125]glucagon specific binding.
Assay data:7 Active, 5 Activity ≤ 1 µM, 7 Tested
IC50 value was expressed for inhibition of [125]glucagon specific binding.
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